Whatsisspharmacodynamics?s-
sCORRECTsANSWER✔whatsasdrugsdoesstosyoursbody
whatsisspharmacokinetics?s-
sCORRECTsANSWER✔whatsyoursbodysdoesstosthesdrug
Thesprocesssofsthesdrugsbeingspreparedstosentersthessystemicscirculation:En
trancesvariessonsthesroutesofsadministration
Includessdrugsmovementsacrossscellsmembranessintosthescirculations-
sCORRECTsANSWER✔absorption
whatsissparentalsabsorptionsroutesmean?s-
sCORRECTsANSWER✔bypasssGIstract
whatsroutescansbeseithersenteralsandsparenteral?s-
sCORRECTsANSWER✔rectal
enteralsisswhatsroutesforsmedsadministration?s-
sCORRECTsANSWER✔oral
whatsroutesofsabsorptionshass100%sbioavailability,sunchangedsandsavailabl
estosbindstosasreceptor.
,Precisesdosing,sEasysaccess,sBolussandscontinuoussdosings-
sCORRECTsANSWER✔IV
Whatsaccountssforsthesfollowingscharacteristics?
sthestimesdelaysbetweenschangessinsplasmasconcentrationsandsdrugseffect.sa
ccountssforsthestimesrequiredsforsdrugstosdiffusesfromsthesplasmastosthessites
ofsactionsplussthestimesrequiredstosillicitsasdrugseffect?s-
sCORRECTsANSWER✔biophase
Whatsroutesissthesonlysroutesthatsdoesn'tspasssthroughsbiologicalsmembrane
s?s-sCORRECTsANSWER✔IV
Thesroutesofsabsorptionsinfluences?s-
sCORRECTsANSWER✔drugsabsorption, sbioavailabity,showsfastsitswork
s
Whatsaresthesabsorptionssitessforsoralsadministration?s-
sCORRECTsANSWER✔smallsintestines(mainly), sstomach,slargesintestin
e
Whatsfactorsfavorssabsorptionsinsansoralsmed?s-
sCORRECTsANSWER✔non-ionized,slipidssoluble,ssmallersmolecules
Whatstypesofsacidsissreadilysabsorbedsbysstomach?s-
sCORRECTsANSWER✔weak
, Weaksacidssmaysbeshighlys________sinsthesalkalinesintestinalspH.
(Thisseffectsisscounterbalancedsbystheslargessurface-
areaseffectsofsthessmallsintestine)s-sCORRECTsANSWER✔ionized
Thesfollowingsdescribesswhatsroute?
sAdvantages:sSustained,stherapeutic splasmaslevels.s
Reducedspeakss/
valleyssassociatedswithsintermittentsdrugsadministration.sAvoidsscontinuo
ussinfusionstechniquesdifficulties.sLowssideseffectsincidences(smallersdoses
).sGenerallysgoodspatientscompliance.s-
sCORRECTsANSWER✔transdermal
Factorsscontributingstosreliables______________sabsorption:s
Molecularsweights<s1000s
pHsranges5s-s9.sNoshistamines-
sreleasingsaction.sDailysdrugsrequirements<s10smg.sUsesofsadjunctsvasoacti
vesdrugs
Epinephrines-sCORRECTsANSWER✔transdermal
whichsrouteshassansunpredictablespharmacologicalsresponse?s-
sCORRECTsANSWER✔rectals(Difficulty sinsprecisesplacement/
sMaysproducesmucosalsirritation)
Whichsrouteshassrapidsandspredictiblesadministrationsroute?
Ensuressactivesdrugsabsorptions
Avoidssfirstspasssmetabolism