Principles of Pharmacology: Pharmacokinetics and Pharmacodynamics: Final exam preparation summary notes 2022
4 Phenotypes of Metabolizers ● UM: Ultrarapid responders ○ Active drugs: ineffective ○ Prodrug: toxic ● EM: Extensive Responders ○ Active drug & prodrug: possibly therapeutic ● IM: Intermediate Responders ○ Active drug & prodrug: possibly therapeutic ● PM: Poor Responders ○ Active drug: toxic ○ Prodrug: ineffective
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